同义名 : | - | |
CAS号 : | 2876918-68-0 | |
货号 : | A1929259 | |
分子式 : | C24H33NO2 | |
纯度 : | 99%+ | |
分子量 : | 367.524 | |
MDL号 : | N/A | |
存储条件: |
粉末 Sealed in dry,Room Temperature 液体 -20°C:3-6个月-80°C:12个月 |
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溶解度 : | - | |
动物实验配方: |
生物活性 | |||
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描述 | CB2R/FAAH modulator-2 is a dual targeting modulator that acts as a CB2R agonist and FAAH inhibitor. CB2R/FAAH modulator-2 possesses Ki values of 10.8 nM and 152.9 nM for CB2R and CB1R, respectively, and an IC50 value of 6.2 μM for FAAH. CB2R/FAAH modulator-2 holds potential for use in studies related to cancer, deleterious inflammatory cascades occurring in neurodegenerative diseases, and COVID-19 infection [1]. |
实验方案 | |||
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1mg | 5mg | 10mg | |
1 mM 5 mM 10 mM |
2.72mL 0.54mL 0.27mL |
13.60mL 2.72mL 1.36mL |
27.21mL 5.44mL 2.72mL |
参考文献 |
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