同义名 : | (S)-MDL100907;(S)-M 100907 | |
CAS号 : | 175673-57-1 | |
货号 : | A1228907 | |
分子式 : | C22H28FNO3 | |
纯度 : | 98%+ | |
分子量 : | 373.461 | |
MDL号 : | MFCD10565916 | |
存储条件: |
粉末 Sealed in dry,2-8°C 液体 -20°C:3-6个月-80°C:12个月 |
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溶解度 : | - | |
动物实验配方: |
生物活性 | |||
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描述 | Volinanserin (MDL 100907) functions as a potent antagonist at the 5-HT2 receptor, displaying a Ki value of 0.36 nM and exhibiting a 300-fold selectivity for the 5-HT2 receptor over the 5-HT1c receptor, alpha-1, and DA D2 receptors. Its activity includes antipsychotic effects[1]. |
实验方案 | |||
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1mg | 5mg | 10mg | |
1 mM 5 mM 10 mM |
2.68mL 0.54mL 0.27mL |
13.39mL 2.68mL 1.34mL |
26.78mL 5.36mL 2.68mL |
参考文献 |
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