生物活性 | |||
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描述 | Ertugliflozin L-pyroglutamic acid (PF-04971729 L-pyroglutamic acid) is a potent, selective, and orally administered inhibitor of the sodium-dependent glucose cotransporter 2 (SGLT2), exhibiting an IC50 of 0.877 nM against h-SGLT2[1]. |
实验方案 | |||
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1mg | 5mg | 10mg | |
1 mM 5 mM 10 mM |
1.77mL 0.35mL 0.18mL |
8.83mL 1.77mL 0.88mL |
17.67mL 3.53mL 1.77mL |
参考文献 |
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